Development of Highly Potent and Selective Covalent FGFR4 Inhibitors Based on SAr Electrophiles Schwarz M, Kurkunov M, Wittlinger F, … Gehringer M · J Med Chem 2024 · J Med Chem 67(8):6549-6569 FGFR4 Tyrosine kinase Covalent inhibitor kineticsInhibitor discovery & SARSelectivity & kinome profiling PhosphoSens Read the paper View on PubMed