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Discovery and characterization of LY2784544, a small-molecule tyrosine kinase inhibitor of JAK2V617F

Ma L, Clayton JR, Walgren RA, … Burkholder TP · Blood Cancer J 2013 · Blood Cancer J 3(4):e109

JAK2 (Tyr) Tyrosine kinase Inhibitor discovery & SARSelectivity & kinome profilingAssay & sensor technology PhosphoSens

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