Selective Inhibitor of Protein Kinase PKN3 Generated by Conjugation of a Structurally Optimized Bumped-(2-Aminoethyl)-8-anilinoisoquinoline-5-sulfonamide (H-9) with d-Arginine-Rich Chain

Smorodina V, Jääger EL, Sõrmus T, … Viht K · Molecules 2026 · Molecules 31(4)

PKN3, PKN1 Ser/Thr kinase Covalent inhibitor kineticsInhibitor discovery & SARSelectivity & kinome profiling PhosphoSens